From: The Hedgehog pathway as targetable vulnerability with 5-azacytidine in myelodysplastic syndrome and acute myeloid leukemia
Cell line
LDE225
GDC0449
EC50 [μM]
MDS-L
15.2
62
TF-1 FLT3-ITD
13.6
–
UKE-1
11.9
HEL
83
ML-2
11.0
12
K562
10.3
32
SET-2
9.7
52
THP-1
9.4
41
OCI-AML3
9.0
38
OCI-AML2
6.9
MV4-11
5.4
M07e
5.2
HL-60
4.3
15
TF-1
3.8
45